La sepiapterina reductasa (SPR) es una enzima que cataliza la reacción final de la síntesis de la tetrahidrobiopterina (BH4) a partir de GTP. Tetrahidrobiopterina + 2 NADP 6-piruvoil-5,6,7,8-tetrahidropterina + 2 NADPH Otras enzimas que participan en la síntesis de la tetrahidrobiopterina son la 6-piruvoiltetrahidropterina sintasa (EC 4.2.3.12) y la GTP ciclohidrolasa I (EC 3.5.4.16).
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